+Search query
-Structure paper
Title | Preclinical evaluation of the SARS-CoV-2 M pro inhibitor RAY1216 shows improved pharmacokinetics compared with nirmatrelvir. |
---|---|
Journal, issue, pages | Nat Microbiol, Vol. 9, Page 1075-1088, Year 2024 |
Publish date | Feb 21, 2023 (structure data deposition date) |
![]() | Chen, X. / Huang, X. / Ma, Q. / Kuzmic, P. / Zhou, B. / Zhang, S. / Chen, J. / Xu, J. / Liu, B. / Jiang, H. ...Chen, X. / Huang, X. / Ma, Q. / Kuzmic, P. / Zhou, B. / Zhang, S. / Chen, J. / Xu, J. / Liu, B. / Jiang, H. / Zhang, W. / Yang, C. / Wu, S. / Huang, J. / Li, H. / Long, C. / Zhao, X. / Xu, H. / Sheng, Y. / Guo, Y. / Niu, C. / Xue, L. / Xu, Y. / Liu, J. / Zhang, T. / Spencer, J. / Zhu, Z. / Deng, W. / Chen, S.H. / Zhong, N. / Xiong, X. / Yang, Z. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2 - 2.02 Å |
Structure data | ![]() PDB-8ign: ![]() PDB-8igo: |
Chemicals | ![]() ChemComp-7ON: ![]() ChemComp-HOH: |
Source |
|
![]() | ![]() ![]() ![]() ![]() ![]() ![]() |