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-Structure paper
Title | Discovery of Aminoratjadone Derivatives as Potent Noncovalent CRM1 Inhibitors. |
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Journal, issue, pages | J. Med. Chem., Vol. 66, Page 11940-11950, Year 2023 |
Publish date | Dec 13, 2022 (structure data deposition date) |
Authors | Jian, L. / Zscherp, R. / Beutling, U. / Shen, X. / Xu, S. / Zhang, X. / Bronstrup, M. / Klahn, P. / Sun, Q. |
External links | J. Med. Chem. / PubMed:37595020 |
Methods | X-ray diffraction |
Resolution | 2.03 - 2.1 Å |
Structure data | PDB-8hq3: PDB-8hq6: |
Chemicals | ChemComp-MG: ChemComp-NO3: ChemComp-GOL: ChemComp-GTP: ChemComp-CL: ChemComp-DMS: ChemComp-MI8: ChemComp-HOH: ChemComp-GLU: ChemComp-MFF: |
Source |
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Keywords | TRANSPORT PROTEIN / nuclear export inhibitor |