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Title | A new generation M pro inhibitor with potent activity against SARS-CoV-2 Omicron variants. |
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Journal, issue, pages | Signal Transduct Target Ther, Vol. 8, Page 128-128, Year 2023 |
Publish date | Nov 17, 2022 (structure data deposition date) |
Authors | Huang, C. / Shuai, H. / Qiao, J. / Hou, Y. / Zeng, R. / Xia, A. / Xie, L. / Fang, Z. / Li, Y. / Yoon, C. ...Huang, C. / Shuai, H. / Qiao, J. / Hou, Y. / Zeng, R. / Xia, A. / Xie, L. / Fang, Z. / Li, Y. / Yoon, C. / Huang, Q. / Hu, B. / You, J. / Quan, B. / Zhao, X. / Guo, N. / Zhang, S. / Ma, R. / Zhang, J. / Wang, Y. / Yang, R. / Nan, J. / Xu, H. / Wang, F. / Lei, J. / Chu, H. / Yang, S. |
External links | Signal Transduct Target Ther / PubMed:36928316 |
Methods | X-ray diffraction |
Resolution | 1.95 - 2.258 Å |
Structure data | PDB-8hht: PDB-8hhu: |
Chemicals | ChemComp-LV0: ChemComp-DMS: ChemComp-HOH: ChemComp-LVX: |
Source |
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Keywords | VIRAL PROTEIN / Severe acute respiratory syndrome coronavirus 2 / main protease |