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-Structure paper
Title | Development of benzimidazole allosteric EGFR kinase inhibitors |
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Journal, issue, pages | To be published |
Publish date | Mar 17, 2023 (structure data deposition date) |
Authors | Beyett, T.S. / Eck, M.J. |
External links | Search PubMed |
Methods | X-ray diffraction |
Resolution | 2.3 Å |
Structure data | PDB-8gk5: |
Chemicals | ChemComp-Q6K:
ChemComp-YW5: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE/INHIBITOR / EGFR / kinase / covalent / inhibitor / allosteric / cancer / TRANSFERASE / TRANSFERASE-INHIBITOR complex |