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-Structure paper
Title | Group 3 medulloblastoma transcriptional networks collapse under domain specific EP300/CBP inhibition. |
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Journal, issue, pages | Nat Commun, Vol. 15, Page 3483-3483, Year 2024 |
Publish date | Jan 18, 2023 (structure data deposition date) |
![]() | Shendy, N.A.M. / Bikowitz, M. / Sigua, L.H. / Zhang, Y. / Mercier, A. / Khashana, Y. / Nance, S. / Liu, Q. / Delahunty, I.M. / Robinson, S. ...Shendy, N.A.M. / Bikowitz, M. / Sigua, L.H. / Zhang, Y. / Mercier, A. / Khashana, Y. / Nance, S. / Liu, Q. / Delahunty, I.M. / Robinson, S. / Goel, V. / Rees, M.G. / Ronan, M.A. / Wang, T. / Kocak, M. / Roth, J.A. / Wang, Y. / Freeman, B.B. / Orr, B.A. / Abraham, B.J. / Roussel, M.F. / Schonbrunn, E. / Qi, J. / Durbin, A.D. |
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Methods | X-ray diffraction |
Resolution | 1.53 - 2.1 Å |
Structure data | ![]() PDB-8fv2: ![]() PDB-8fvf: ![]() PDB-8fvk: ![]() PDB-8fvs: ![]() PDB-8fxa: ![]() PDB-8fxe: ![]() PDB-8fxo: ![]() PDB-8g6t: ![]() PDB-8ga2: |
Chemicals | ![]() ChemComp-PO4: ![]() ChemComp-JHL: ![]() ChemComp-EDO: ![]() ChemComp-HOH: ![]() ChemComp-NI: ![]() ChemComp-SO4: ![]() ChemComp-YBE: ![]() ChemComp-MG: ![]()
ChemComp-YJY: ![]()
ChemComp-YID: ![]()
ChemComp-YN5: ![]()
ChemComp-YRI: ![]()
ChemComp-YVK: |
Source |
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![]() | TRANSCRIPTION/INHIBITOR / bromodomain / small molecule ligand / complex / TRANSCRIPTION / TRANSCRIPTION-INHIBITOR complex / TRANSFERASE / TRANSFERASE/TRANSFERASE INHIBITOR / TRANSFERASE-TRANSFERASE INHIBITOR complex |