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-Structure paper
Title | Exploring Covalent Bond Formation at Tyr-82 for Inhibition of Ral GTPase Activation. |
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Journal, issue, pages | Chemmedchem, Vol. 18, Page e202300272-e202300272, Year 2023 |
Publish date | Dec 19, 2022 (structure data deposition date) |
![]() | Landgraf, A.D. / Yeh, I.J. / Ghozayel, M.K. / Bum-Erdene, K. / Gonzalez-Gutierrez, G. / Meroueh, S.O. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.48 - 1.54 Å |
Structure data | ![]() PDB-8fjh: ![]() PDB-8fji: |
Chemicals | ![]() ChemComp-GDP: ![]() ChemComp-Y0P: ![]() ChemComp-CA: ![]() ChemComp-HOH: ![]() ChemComp-Y0M: |
Source |
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![]() | HYDROLASE/HYDROLASE INHIBITOR / RalA / GTPase / inhibitor / HYDROLASE / HYDROLASE-HYDROLASE INHIBITOR complex |