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-Structure paper
Title | Discovery and Characterization of Potent, Efficacious, Orally Available Antimalarial Plasmepsin X Inhibitors and Preclinical Safety Assessment of UCB7362 . |
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Journal, issue, pages | J. Med. Chem., Vol. 65, Page 14121-14143, Year 2022 |
Publish date | Jul 22, 2022 (structure data deposition date) |
![]() | Lowe, M.A. / Cardenas, A. / Valentin, J.P. / Zhu, Z. / Abendroth, J. / Castro, J.L. / Class, R. / Delaunois, A. / Fleurance, R. / Gerets, H. ...Lowe, M.A. / Cardenas, A. / Valentin, J.P. / Zhu, Z. / Abendroth, J. / Castro, J.L. / Class, R. / Delaunois, A. / Fleurance, R. / Gerets, H. / Gryshkova, V. / King, L. / Lorimer, D.D. / MacCoss, M. / Rowley, J.H. / Rosseels, M.L. / Royer, L. / Taylor, R.D. / Wong, M. / Zaccheo, O. / Chavan, V.P. / Ghule, G.A. / Tapkir, B.K. / Burrows, J.N. / Duffey, M. / Rottmann, M. / Wittlin, S. / Angulo-Barturen, I. / Jimenez-Diaz, M.B. / Striepen, J. / Fairhurst, K.J. / Yeo, T. / Fidock, D.A. / Cowman, A.F. / Favuzza, P. / Crespo-Fernandez, B. / Gamo, F.J. / Goldberg, D.E. / Soldati-Favre, D. / Laleu, B. / de Haro, T. |
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Methods | X-ray diffraction |
Resolution | 2.85 Å |
Structure data | ![]() PDB-8dsr: |
Chemicals | ![]() ChemComp-TWU: |
Source |
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![]() | HYDROLASE / Plasmepsin X / Plasmodium falciparum / PM10 / PMX |