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Title | Biolayer Interferometry Assay for Cyclin-Dependent Kinase-Cyclin Association Reveals Diverse Effects of Cdk2 Inhibitors on Cyclin Binding Kinetics. |
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Journal, issue, pages | Acs Chem. Biol., Vol. 18, Page 431-440, Year 2023 |
Publish date | May 17, 2022 (structure data deposition date) |
Authors | Tambo, C.S. / Tripathi, S. / Perera, B.G.K. / Maly, D.J. / Bridges, A.J. / Kiss, G. / Rubin, S.M. |
External links | Acs Chem. Biol. / PubMed:36724382 |
Methods | X-ray diffraction |
Resolution | 2.2 Å |
Structure data | PDB-8cur: |
Chemicals | ChemComp-OW6: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE/INHIBITOR / cell cycle / protein-inhibitor complex / kinase / TRANSFERASE-INHIBITOR complex |