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-Structure paper
Title | Selective Wee1 Inhibitors Led to Antitumor Activity In Vitro and Correlated with Myelosuppression. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 14, Page 566-576, Year 2023 |
Publish date | Nov 6, 2022 (structure data deposition date) |
![]() | Guler, S. / DiPoto, M.C. / Crespo, A. / Caldwell, R. / Doerfel, B. / Grossmann, N. / Ho, K. / Huck, B. / Jones, C.C. / Lan, R. ...Guler, S. / DiPoto, M.C. / Crespo, A. / Caldwell, R. / Doerfel, B. / Grossmann, N. / Ho, K. / Huck, B. / Jones, C.C. / Lan, R. / Musil, D. / Potnick, J. / Schilke, H. / Sherer, B. / Simon, S. / Sirrenberg, C. / Zhang, Z. / Liu-Bujalski, L. |
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Methods | X-ray diffraction |
Resolution | 1.53 - 2.188 Å |
Structure data | ![]() PDB-8bjt: ![]() PDB-8bju: |
Chemicals | ![]() ChemComp-ACT: ![]() ChemComp-8X7: ![]() ChemComp-ZN: ![]() ChemComp-HOH: ![]() ChemComp-QT9: |
Source |
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![]() | TRANSFERASE / PLK1 / SELECTIVITY RESIDUES / KINASE / POLO-LIKE KINASE / STRUCTURE BASED DRUG DESIGN / ATP-BINDING / NUCLEOTIDE-BINDING / PHOSPHORYLATION / SERINE/THREONINE-PROTEIN KINASE / WEE1 / PROTEIN-INHIBITOR COMPLEX |