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-Structure paper
Title | Discovery, Characterization, and Structure-Based Optimization of Small-Molecule In Vitro and In Vivo Probes for Human DNA Polymerase Theta. |
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Journal, issue, pages | J. Med. Chem., Vol. 65, Page 13879-13891, Year 2022 |
Publish date | May 13, 2022 (structure data deposition date) |
![]() | Stockley, M.L. / Ferdinand, A. / Benedetti, G. / Blencowe, P. / Boyd, S.M. / Calder, M. / Charles, M.D. / Edwardes, L.V. / Ekwuru, T. / Finch, H. ...Stockley, M.L. / Ferdinand, A. / Benedetti, G. / Blencowe, P. / Boyd, S.M. / Calder, M. / Charles, M.D. / Edwardes, L.V. / Ekwuru, T. / Finch, H. / Galbiati, A. / Geo, L. / Grande, D. / Grinkevich, V. / Holliday, N.D. / Krajewski, W.W. / MacDonald, E. / Majithiya, J.B. / McCarron, H. / McWhirter, C.L. / Patel, V. / Pedder, C. / Rajendra, E. / Ranzani, M. / Rigoreau, L.J.M. / Robinson, H.M.R. / Schaedler, T. / Sirina, J. / Smith, G.C.M. / Swarbrick, M.E. / Turnbull, A.P. / Willis, S. / Heald, R.A. |
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Methods | X-ray diffraction |
Resolution | 2.26 - 2.99 Å |
Structure data | ![]() PDB-7zus: ![]() PDB-7zx0: ![]() PDB-7zx1: |
Chemicals | ![]() ChemComp-MG: ![]() ChemComp-DG3: ![]() ChemComp-HOH: ![]() ChemComp-K7X: ![]() ChemComp-K8I: |
Source |
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![]() | TRANSFERASE / DNA polymerase / protein-DNA complex / DNA repair / inhibitor |