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-Structure paper
Title | Substrate-Based Design of Cytosolic Nucleotidase IIIB Inhibitors and Structural Insights into Inhibition Mechanism. |
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Journal, issue, pages | Pharmaceuticals, Vol. 15, Year 2022 |
Publish date | Mar 31, 2022 (structure data deposition date) |
![]() | Kubacka, D. / Kozarski, M. / Baranowski, M.R. / Wojcik, R. / Panecka-Hofman, J. / Strzelecka, D. / Basquin, J. / Jemielity, J. / Kowalska, J. |
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Methods | X-ray diffraction |
Resolution | 1.36 - 1.56 Å |
Structure data | ![]() PDB-7zee: ![]() PDB-7zeg: ![]() PDB-7zeh: |
Chemicals | ![]() ChemComp-MES: ![]() ChemComp-MG: ![]() ChemComp-EDO: ![]() ChemComp-HOH: ![]() ChemComp-IOO: ![]() ChemComp-IPQ: ![]() ChemComp-RBL: ![]() ChemComp-PO4: ![]() ChemComp-SO4: |
Source |
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![]() | HYDROLASE / cytosolic 5' nucleotidase / N7 methylguanosine monophosphate dephosphorylation / mRNA cap degradation / nucleotide level regulation |