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-Structure paper
Title | Discovery of novel covalent selective estrogen receptor degraders against endocrine-resistant breast cancer. |
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Journal, issue, pages | Acta Pharm Sin B, Vol. 13, Page 4963-4982, Year 2023 |
Publish date | Jul 28, 2022 (structure data deposition date) |
![]() | Wang, Y. / Min, J. / Deng, X. / Feng, T. / Hu, H. / Guo, X. / Cheng, Y. / Xie, B. / Yang, Y. / Chen, C.C. ...Wang, Y. / Min, J. / Deng, X. / Feng, T. / Hu, H. / Guo, X. / Cheng, Y. / Xie, B. / Yang, Y. / Chen, C.C. / Guo, R.T. / Dong, C. / Zhou, H.B. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.25 Å |
Structure data | ![]() PDB-7ymk: |
Chemicals | ![]() ChemComp-PEG: ![]() ChemComp-IX0: ![]() ChemComp-SO4: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSCRIPTION/INHIBITOR / Complex / Inhibitor / Estrogen Receptor Alpha / TRANSCRIPTION-INHIBITOR complex / TRANSCRIPTION |