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Title | Discovery of BGB-8035, a Highly Selective Covalent Inhibitor of Bruton's Tyrosine Kinase for B-Cell Malignancies and Autoimmune Diseases. |
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Journal, issue, pages | J. Med. Chem., Vol. 66, Page 4025-4044, Year 2023 |
Publish date | Jul 1, 2022 (structure data deposition date) |
Authors | Guo, Y. / Hu, N. / Liu, Y. / Zhang, W. / Yu, D. / Shi, G. / Zhang, B. / Yin, L. / Wei, M. / Yuan, X. ...Guo, Y. / Hu, N. / Liu, Y. / Zhang, W. / Yu, D. / Shi, G. / Zhang, B. / Yin, L. / Wei, M. / Yuan, X. / Luo, L. / Wang, F. / Song, X. / Xin, L. / Wei, Q. / Li, Y. / Chen, S. / Zhang, T. / Zhang, S. / Zhou, X. / Zhang, C. / Su, D. / Liu, J. / Cheng, Z. / Zhang, J. / Xing, H. / Sun, H. / Li, X. / Zhao, Y. / He, M. / Wu, Y. / Sun, X. / Tian, A. / Zhou, C. / Young, S. / Liu, X. / Wang, L. / Wang, Z. |
External links | J. Med. Chem. / PubMed:36912866 |
Methods | X-ray diffraction |
Resolution | 1.4 Å |
Structure data | PDB-7yc9: |
Chemicals | ChemComp-IS4: ChemComp-EDO: ChemComp-HOH: |
Source |
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Keywords | ANTITUMOR PROTEIN / kinase / inhibitor / complex |