+Search query
-Structure paper
Title | Characterization of the cholangiocarcinoma drug pemigatinib against FGFR gatekeeper mutants. |
---|---|
Journal, issue, pages | Commun Chem, Vol. 5, Page 100-100, Year 2022 |
Publish date | Dec 20, 2021 (structure data deposition date) |
Authors | Lin, Q. / Chen, X. / Qu, L. / Guo, M. / Wei, H. / Dai, S. / Jiang, L. / Chen, Y. |
External links | Commun Chem / PubMed:36698015 |
Methods | X-ray diffraction |
Resolution | 2.495 Å |
Structure data | PDB-7wcl: |
Chemicals | ChemComp-8ZF: ChemComp-SO4: ChemComp-HOH: |
Source |
|
Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / Kinase / Inhibitor / Complex / STRUCTURAL PROTEIN / TRANSFERASE-TRANSFERASE INHIBITOR complex / TRA |