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-Structure paper
Title | Fragment-Based Discovery of AF9 YEATS Domain Inhibitors. |
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Journal, issue, pages | Int J Mol Sci, Vol. 23, Year 2022 |
Publish date | Sep 29, 2021 (structure data deposition date) |
Authors | Liu, Y. / Jin, R. / Lu, H. / Bian, K. / Wang, R. / Wang, L. / Gao, R. / Zhang, J. / Wu, J. / Yao, X. ...Liu, Y. / Jin, R. / Lu, H. / Bian, K. / Wang, R. / Wang, L. / Gao, R. / Zhang, J. / Wu, J. / Yao, X. / Liu, X. / Liu, D. / Wang, X. / Zhang, Z. / Ruan, K. |
External links | Int J Mol Sci / PubMed:35409252 |
Methods | X-ray diffraction |
Resolution | 1.83 - 2.25 Å |
Structure data | PDB-7vkg: PDB-7vkh: |
Chemicals | ChemComp-7IV: ChemComp-CL: ChemComp-EDO: ChemComp-HOH: ChemComp-7IY: ChemComp-GOL: |
Source |
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Keywords | TRANSCRIPTION / Complex / inhibitor |