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-Structure paper
Title | Discovery of 10H-Benzo[b]pyrido[2,3-e][1,4]oxazine AXL Inhibitors via Structure-Based Drug Design Targeting c-Met Kinase |
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Journal, issue, pages | J. Med. Chem., Vol. 66, Page 220-234, Year 2023 |
Publish date | Aug 11, 2021 (structure data deposition date) |
![]() | Zhan, Z. / Ji, Y. / Su, H. / Fang, C. / Peng, X. / Liu, Q. / Dai, Y. / Lin, D. / Xu, Y. / Ai, J. / Duan, W. |
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Methods | X-ray diffraction |
Resolution | 1.7 - 1.9 Å |
Structure data | ![]() PDB-7v3r: ![]() PDB-7v3s: |
Chemicals | ![]() ChemComp-5IE: ![]() ChemComp-HOH: ![]() ChemComp-5I9: |
Source |
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![]() | TRANSFERASE/INHIBITOR / TRANSFERASE-INHIBITOR COMPLEX |