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-Structure paper
Title | ATP-site inhibitors induce unique conformations of the acute myeloid leukemia-associated Src-family kinase, Fgr. |
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Journal, issue, pages | Structure, Vol. 30, Page 1508-1517.e3, Year 2022 |
Publish date | May 6, 2022 (structure data deposition date) |
![]() | Du, S. / Alvarado, J.J. / Wales, T.E. / Moroco, J.A. / Engen, J.R. / Smithgall, T.E. |
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Methods | X-ray diffraction |
Resolution | 2.55 - 2.99 Å |
Structure data | ![]() PDB-7uy0: ![]() PDB-7uy3: |
Chemicals | ![]() ChemComp-GOL: ![]() ChemComp-VSE: ![]() ChemComp-CL: ![]() ChemComp-PO4: ![]() ChemComp-HOH: ![]() ChemComp-OJL: ![]() ChemComp-EDO: |
Source |
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![]() | TRANSFERASE / Fgr / A-419259 / SIGNALING PROTEIN / kinase / TL02-59 |