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Title1,4-Dihydropyridinebutyrolactone-derived ring-opened ester and amide analogs targeting BET bromodomains.
Journal, issue, pagesArch Pharm, Vol. 355, Page e2200288-e2200288, Year 2022
Publish dateApr 28, 2022 (structure data deposition date)
AuthorsJiang, J. / Zhao, P.L. / Sigua, L.H. / Chan, A. / Schonbrunn, E. / Qi, J. / Georg, G.I.
External linksArch Pharm / PubMed:35941525
MethodsX-ray diffraction
Resolution1.52 - 1.55 Å
Structure data

PDB-7uty:
First bromodomain of BRD4 liganded with compound 2c
Method: X-RAY DIFFRACTION / Resolution: 1.55 Å

PDB-7uuu:
First bromodomain of BRDT liganded with compound 2c
Method: X-RAY DIFFRACTION / Resolution: 1.52 Å

Chemicals

ChemComp-OFR:
prop-2-en-1-yl (5S)-1-ethyl-7-methyl-5-(4-methylphenyl)-2,4-dioxo-1,2,3,4,5,8-hexahydropyrido[2,3-d]pyrimidine-6-carboxylate

ChemComp-EDO:
1,2-ETHANEDIOL

ChemComp-HOH:
WATER

Source
  • homo sapiens (human)
KeywordsTRANSCRIPTION / Inhibitor / acetyl-lysine / transcription regulation

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