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-Structure paper
Title | Repurposed dihydroorotate dehydrogenase inhibitors with efficacy against drug-resistant Acinetobacter baumannii. |
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Journal, issue, pages | Proc. Natl. Acad. Sci. USA, Vol. 119, Page e2213116119-e2213116119, Year 2022 |
Publish date | Apr 26, 2022 (structure data deposition date) |
Authors | Russo, T.A. / Umland, T.C. / Deng, X. / El Mazouni, F. / Kokkonda, S. / Olson, R. / Carlino-MacDonald, U. / Beanan, J. / Alvarado, C.L. / Tomchick, D.R. ...Russo, T.A. / Umland, T.C. / Deng, X. / El Mazouni, F. / Kokkonda, S. / Olson, R. / Carlino-MacDonald, U. / Beanan, J. / Alvarado, C.L. / Tomchick, D.R. / Hutson, A. / Chen, H. / Posner, B. / Rathod, P.K. / Charman, S.A. / Phillips, M.A. |
External links | Proc. Natl. Acad. Sci. USA / PubMed:36512492 |
Methods | X-ray diffraction |
Resolution | 1.4 Å |
Structure data | PDB-7ut5: |
Chemicals | ChemComp-OBR: ChemComp-FMN: ChemComp-ORO: ChemComp-GOL: ChemComp-HOH: |
Source |
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Keywords | OXIDOREDUCTASE/INHIBITOR / inhibitor / complex / Flavoprotein / OXIDOREDUCTASE / OXIDOREDUCTASE-INHIBITOR complex |