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-Structure paper
Title | GRL-142 binds to and impairs HIV-1 integrase nuclear localization signal and potently suppresses highly INSTI-resistant HIV-1 variants. |
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Journal, issue, pages | Sci Adv, Vol. 9, Page eadg2955-eadg2955, Year 2023 |
Publish date | Mar 21, 2022 (structure data deposition date) |
![]() | Aoki, M. / Aoki-Ogata, H. / Bulut, H. / Hayashi, H. / Takamune, N. / Kishimoto, N. / Tanaka, H. / Higashi-Kuwata, N. / Hattori, S.I. / Das, D. ...Aoki, M. / Aoki-Ogata, H. / Bulut, H. / Hayashi, H. / Takamune, N. / Kishimoto, N. / Tanaka, H. / Higashi-Kuwata, N. / Hattori, S.I. / Das, D. / Venkateswara Rao, K. / Iwama, K. / Davis, D.A. / Hasegawa, K. / Murayama, K. / Yarchoan, R. / Ghosh, A.K. / Pau, A.K. / Machida, S. / Misumi, S. / Mitsuya, H. |
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Methods | X-ray diffraction |
Resolution | 3 Å |
Structure data | ![]() PDB-7ue1: |
Chemicals | ![]() ChemComp-7OA: ![]() ChemComp-SO4: |
Source |
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![]() | VIRAL PROTEIN / Inhibitor |