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-Structure paper
Title | 1,3-Diarylpyrazolyl-acylsulfonamides Target HadAB/BC Complex in Mycobacterium tuberculosis . |
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Journal, issue, pages | Acs Infect Dis., Vol. 8, Page 2315-2326, Year 2022 |
Publish date | Nov 19, 2021 (structure data deposition date) |
![]() | Singh, V. / Grzegorzewicz, A.E. / Fienberg, S. / Muller, R. / Khonde, L.P. / Sanz, O. / Alfonso, S. / Urones, B. / Drewes, G. / Bantscheff, M. ...Singh, V. / Grzegorzewicz, A.E. / Fienberg, S. / Muller, R. / Khonde, L.P. / Sanz, O. / Alfonso, S. / Urones, B. / Drewes, G. / Bantscheff, M. / Ghidelli-Disse, S. / Ioerger, T.R. / Angala, B. / Liu, J. / Lee, R.E. / Sacchettini, J.C. / Krieger, I.V. / Jackson, M. / Chibale, K. / Ghorpade, S.R. |
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Methods | X-ray diffraction |
Resolution | 2.4 Å |
Structure data | ![]() PDB-7svt: |
Chemicals | ![]() ChemComp-CI7: ![]() ChemComp-EDO: ![]() ChemComp-PEG: ![]() ChemComp-GOL: ![]() ChemComp-HOH: |
Source |
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![]() | LYASE/INHIBITOR / Mycobacterium tuberculosis / Tuberculosis drug discovery / 3-hydroxyl-ACP dehydratase / HadAB/BC / Structural Genomics / TB Structural Genomics Consortium / TBSGC / lipid binding protein / LYASE-INHIBITOR complex |