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-Structure paper
Title | Discovery of Non-Nucleotide Small-Molecule STING Agonists via Chemotype Hybridization. |
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Journal, issue, pages | J. Med. Chem., Vol. 65, Page 3518-3538, Year 2022 |
Publish date | Nov 11, 2021 (structure data deposition date) |
Authors | Cherney, E.C. / Zhang, L. / Lo, J. / Huynh, T. / Wei, D. / Ahuja, V. / Quesnelle, C. / Schieven, G.L. / Futran, A. / Locke, G.A. ...Cherney, E.C. / Zhang, L. / Lo, J. / Huynh, T. / Wei, D. / Ahuja, V. / Quesnelle, C. / Schieven, G.L. / Futran, A. / Locke, G.A. / Lin, Z. / Monereau, L. / Chaudhry, C. / Blum, J. / Li, S. / Fereshteh, M. / Li-Wang, B. / Gangwar, S. / Pan, C. / Chong, C. / Zhu, X. / Posy, S.L. / Sack, J.S. / Zhang, P. / Ruzanov, M. / Harner, M. / Akhtar, F. / Schroeder, G.M. / Vite, G. / Fink, B. |
External links | J. Med. Chem. / PubMed:35108011 |
Methods | X-ray diffraction |
Resolution | 1.96 Å |
Structure data | PDB-7ssm: |
Chemicals | ChemComp-B7L: ChemComp-HOH: |
Source |
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Keywords | IMMUNE SYSTEM / RECEPTOR |