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-Structure paper
Title | PPAR gamma Corepression Involves Alternate Ligand Conformation and Inflation of H12 Ensembles. |
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Journal, issue, pages | Acs Chem. Biol., Vol. 18, Page 1115-1123, Year 2023 |
Publish date | Nov 5, 2021 (structure data deposition date) |
Authors | Frkic, R.L. / Pederick, J.L. / Horsfall, A.J. / Jovcevski, B. / Crame, E.E. / Kowalczyk, W. / Pukala, T.L. / Chang, M.R. / Zheng, J. / Blayo, A.L. ...Frkic, R.L. / Pederick, J.L. / Horsfall, A.J. / Jovcevski, B. / Crame, E.E. / Kowalczyk, W. / Pukala, T.L. / Chang, M.R. / Zheng, J. / Blayo, A.L. / Abell, A.D. / Kamenecka, T.M. / Harbort, J.S. / Harmer, J.R. / Griffin, P.R. / Bruning, J.B. |
External links | Acs Chem. Biol. / PubMed:37146157 |
Methods | X-ray diffraction |
Resolution | 2.499 - 2.6 Å |
Structure data | PDB-7sqa: PDB-7sqb: |
Chemicals | ChemComp-A8R: ChemComp-HOH: |
Source |
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Keywords | TRANSCRIPTION / Inverse agonist / Nuclear receptor / Ligand binding domain / corepressor / Helix 12 |