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Title | Discovery of Inhibitors of the Lipopolysaccharide Transporter MsbA: From a Screening Hit to Potent Wild-Type Gram-Negative Activity. |
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Journal, issue, pages | J. Med. Chem., Vol. 65, Page 4085-4120, Year 2022 |
Publish date | Sep 30, 2021 (structure data deposition date) |
Authors | Verma, V.A. / Wang, L. / Labadie, S.S. / Liang, J. / Sellers, B.D. / Wang, J. / Dong, L. / Wang, Q. / Zhang, S. / Xu, Z. ...Verma, V.A. / Wang, L. / Labadie, S.S. / Liang, J. / Sellers, B.D. / Wang, J. / Dong, L. / Wang, Q. / Zhang, S. / Xu, Z. / Zhang, Y. / Niu, Y. / Wang, X. / Wai, J. / Koehler, M.F.T. / Hu, H. / Alexander, M.K. / Nishiyama, M. / Miu, A. / Xu, Y. / Pang, J. / Katakam, A.K. / Reichelt, M. / Austin, C.D. / Ho, H. / Payandeh, J. / Koth, C.M. |
External links | J. Med. Chem. / PubMed:35184554 |
Methods | X-ray diffraction |
Resolution | 2.978 Å |
Structure data | PDB-7sel: |
Chemicals | ChemComp-95X: ChemComp-KDL: |
Source |
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Keywords | TRANSLOCASE / MsbA / Lipid A / LPS / inhibitor / LIPID TRANSPORT |