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-Structure paper
Title | Crystal structure of the first bromodomain (BD1) of human BRD4 in complex with dual BRD4-JAK2 inhibitor MA9-086 |
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Journal, issue, pages | To Be Published |
Publish date | Jul 13, 2021 (structure data deposition date) |
![]() | Karim, M.R. / Schonbrunn, E. |
![]() | Search PubMed |
Methods | X-ray diffraction |
Resolution | 1.2 Å |
Structure data | ![]() PDB-7rek: |
Chemicals | ![]() ChemComp-R6S: ![]() ChemComp-EDO: ![]() ChemComp-HOH: |
Source |
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![]() | GENE REGULATION / BET / JAK2 / dual BRD-kinase inhibitor |