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-Structure paper
Title | Discovery of SY-5609: A Selective, Noncovalent Inhibitor of CDK7. |
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Journal, issue, pages | J. Med. Chem., Vol. 65, Page 1458-1480, Year 2022 |
Publish date | Jun 30, 2021 (structure data deposition date) |
![]() | Marineau, J.J. / Hamman, K.B. / Hu, S. / Alnemy, S. / Mihalich, J. / Kabro, A. / Whitmore, K.M. / Winter, D.K. / Roy, S. / Ciblat, S. ...Marineau, J.J. / Hamman, K.B. / Hu, S. / Alnemy, S. / Mihalich, J. / Kabro, A. / Whitmore, K.M. / Winter, D.K. / Roy, S. / Ciblat, S. / Ke, N. / Savinainen, A. / Wilsily, A. / Malojcic, G. / Zahler, R. / Schmidt, D. / Bradley, M.J. / Waters, N.J. / Chuaqui, C. |
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Methods | X-ray diffraction |
Resolution | 1.67 Å |
Structure data | ![]() PDB-7ra5: |
Chemicals | ![]() ChemComp-3I3: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE/INHIBITOR / CDK2 / CYCLIN-DEPENDENT KINASE 2 / PROTEROS BIOSTRUCTURES GMBH / TRANSFERASE / TRANSFERASE-INHIBITOR complex |