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| Title | Chemical Optimization of Selective Pseudomonas aeruginosa LasB Elastase Inhibitors and Their Impact on LasB-Mediated Activation of IL-1 beta in Cellular and Animal Infection Models. |
|---|---|
| Journal, issue, pages | Acs Infect Dis., Vol. 9, Page 270-282, Year 2023 |
| Publish date | Dec 10, 2021 (structure data deposition date) |
Authors | Everett, M.J. / Davies, D.T. / Leiris, S. / Sprynski, N. / Llanos, A. / Castandet, J.M. / Lozano, C. / LaRock, C.N. / LaRock, D.L. / Corsica, G. ...Everett, M.J. / Davies, D.T. / Leiris, S. / Sprynski, N. / Llanos, A. / Castandet, J.M. / Lozano, C. / LaRock, C.N. / LaRock, D.L. / Corsica, G. / Docquier, J.D. / Pallin, T.D. / Cridland, A. / Blench, T. / Zalacain, M. / Lemonnier, M. |
External links | Acs Infect Dis. / PubMed:36669138 |
| Methods | X-ray diffraction |
| Resolution | 2.74 Å |
| Structure data | ![]() PDB-7qh1: |
| Chemicals | ![]() ChemComp-ZN: ![]() ChemComp-CI8: ![]() ChemComp-CA: ![]() ChemComp-HOH: |
| Source |
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Keywords | HYDROLASE / Pseudomonas aeruginosa / respiratory disease |
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