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-Structure paper
Title | Identification and optimisation of a pyrimidopyridone series of IRAK4 inhibitors. |
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Journal, issue, pages | Bioorg. Med. Chem., Vol. 63, Page 116729-116729, Year 2022 |
Publish date | Dec 7, 2021 (structure data deposition date) |
![]() | Cumming, I.A. / Degorce, S.L. / Aagaard, A. / Braybrooke, E.L. / Davies, N.L. / Diene, C.R. / Eatherton, A.J. / Felstead, H.R. / Groombridge, S.D. / Lenz, E.M. ...Cumming, I.A. / Degorce, S.L. / Aagaard, A. / Braybrooke, E.L. / Davies, N.L. / Diene, C.R. / Eatherton, A.J. / Felstead, H.R. / Groombridge, S.D. / Lenz, E.M. / Li, Y. / Nai, Y. / Pearson, S. / Robb, G.R. / Scott, J.S. / Steward, O.R. / Wu, C. / Xue, Y. / Zhang, L. / Zhang, Y. |
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Methods | X-ray diffraction |
Resolution | 2.07 - 3.031 Å |
Structure data | ![]() PDB-7qg1: ![]() PDB-7qg2: ![]() PDB-7qg3: ![]() PDB-7qg5: |
Chemicals | ![]() ChemComp-B8I: ![]() ChemComp-HOH: ![]() ChemComp-B6I: ![]() ChemComp-B4U: ![]() ChemComp-B7R: |
Source |
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![]() | TRANSFERASE / Kinase inhibitor Interleukin-1 Receptor-Associated Kinase 4 Interleukin-1 signaling |