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-Structure paper
Title | Structure-Based Design of Dual Partial Peroxisome Proliferator-Activated Receptor gamma Agonists/Soluble Epoxide Hydrolase Inhibitors. |
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Journal, issue, pages | J. Med. Chem., Vol. 64, Page 17259-17276, Year 2021 |
Publish date | Jul 11, 2021 (structure data deposition date) |
Authors | Lillich, F.F. / Willems, S. / Ni, X. / Kilu, W. / Borkowsky, C. / Brodsky, M. / Kramer, J.S. / Brunst, S. / Hernandez-Olmos, V. / Heering, J. ...Lillich, F.F. / Willems, S. / Ni, X. / Kilu, W. / Borkowsky, C. / Brodsky, M. / Kramer, J.S. / Brunst, S. / Hernandez-Olmos, V. / Heering, J. / Schierle, S. / Kestner, R.I. / Mayser, F.M. / Helmstadter, M. / Gobel, T. / Weizel, L. / Namgaladze, D. / Kaiser, A. / Steinhilber, D. / Pfeilschifter, W. / Kahnt, A.S. / Proschak, A. / Chaikuad, A. / Knapp, S. / Merk, D. / Proschak, E. |
External links | J. Med. Chem. / PubMed:34818007 |
Methods | X-ray diffraction |
Resolution | 2.15 - 2.4 Å |
Structure data | PDB-7p4e: PDB-7p4k: |
Chemicals | ChemComp-5IV: ChemComp-SO4: ChemComp-EDO: ChemComp-HOH: |
Source |
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Keywords | DNA BINDING PROTEIN / complex / Structural Genomics / Structural Genomics Consortium / SGC / HYDROLASE |