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-Structure paper
Title | Identification of Pyrimidine-Based Lead Compounds for Understudied Kinases Implicated in Driving Neurodegeneration. |
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Journal, issue, pages | J. Med. Chem., Vol. 65, Page 1313-1328, Year 2022 |
Publish date | Jul 1, 2021 (structure data deposition date) |
Authors | Drewry, D.H. / Annor-Gyamfi, J.K. / Wells, C.I. / Pickett, J.E. / Dederer, V. / Preuss, F. / Mathea, S. / Axtman, A.D. |
External links | J. Med. Chem. / PubMed:34333981 |
Methods | X-ray diffraction |
Resolution | 1.95 Å |
Structure data | PDB-7p1l: |
Chemicals | ChemComp-V5E: ChemComp-EDO: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE / Kinase Inhibitor Active site Folded activation loop UBA domain |