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-Structure paper
Title | Pyridylpiperazine-based allosteric inhibitors of RND-type multidrug efflux pumps. |
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Journal, issue, pages | Nat Commun, Vol. 13, Page 115-115, Year 2022 |
Publish date | Jun 12, 2021 (structure data deposition date) |
![]() | Ple, C. / Tam, H.K. / Vieira Da Cruz, A. / Compagne, N. / Jimenez-Castellanos, J.C. / Muller, R.T. / Pradel, E. / Foong, W.E. / Malloci, G. / Ballee, A. ...Ple, C. / Tam, H.K. / Vieira Da Cruz, A. / Compagne, N. / Jimenez-Castellanos, J.C. / Muller, R.T. / Pradel, E. / Foong, W.E. / Malloci, G. / Ballee, A. / Kirchner, M.A. / Moshfegh, P. / Herledan, A. / Herrmann, A. / Deprez, B. / Willand, N. / Vargiu, A.V. / Pos, K.M. / Flipo, M. / Hartkoorn, R.C. |
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Methods | X-ray diffraction |
Resolution | 2.45 - 2.8 Å |
Structure data | ![]() PDB-7ouk: ![]() PDB-7oul: ![]() PDB-7oum: |
Chemicals | ![]() ChemComp-LMT: ![]() ChemComp-1K8: ![]() ChemComp-EDO: ![]() ChemComp-OCT: ![]() ChemComp-C14: ![]() ChemComp-GOL: ![]() ChemComp-D10: ![]() ChemComp-DDR: ![]() ChemComp-DDQ: ![]() ChemComp-SO4: ![]() ChemComp-LPX: ![]() ChemComp-HOH: ![]() ChemComp-1KE: ![]() ChemComp-D12: |
Source |
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![]() | TRANSPORT PROTEIN / Multidrug efflux pump / Membrane protein |