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-Structure paper
Title | Interrogating the Inhibition Mechanisms of Human Aldehyde Oxidase by X-ray Crystallography and NMR Spectroscopy: The Raloxifene Case. |
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Journal, issue, pages | J. Med. Chem., Vol. 64, Page 13025-13037, Year 2021 |
Publish date | Jun 1, 2021 (structure data deposition date) |
![]() | Mota, C. / Diniz, A. / Coelho, C. / Santos-Silva, T. / Esmaeeli, M. / Leimkuhler, S. / Cabrita, E.J. / Marcelo, F. / Romao, M.J. |
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Methods | X-ray diffraction |
Resolution | 2.6 - 2.7 Å |
Structure data | ![]() PDB-7opn: ![]() PDB-7orc: |
Chemicals | ![]() ChemComp-FES: ![]() ChemComp-MTE: ![]() ChemComp-MOS: ![]() ChemComp-FAD: ![]() ChemComp-MLI: ![]() ChemComp-PG6: ![]() ChemComp-GOL: ![]() ChemComp-RAL: ![]() ChemComp-DMS: ![]() ChemComp-HOH: |
Source |
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![]() | OXIDOREDUCTASE / Human Aldehyde Oxidase / Single Nucleotide Polymorphism / Complex / Inhibitor |