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-Structure paper
Title | Crystal Structure-Guided Design of Bisubstrate Inhibitors and Photoluminescent Probes for Protein Kinases of the PIM Family. |
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Journal, issue, pages | Molecules, Vol. 26, Year 2021 |
Publish date | May 28, 2021 (structure data deposition date) |
Authors | Nonga, O.E. / Lavogina, D. / Enkvist, E. / Kestav, K. / Chaikuad, A. / Dixon-Clarke, S.E. / Bullock, A.N. / Kopanchuk, S. / Ivan, T. / Ekambaram, R. ...Nonga, O.E. / Lavogina, D. / Enkvist, E. / Kestav, K. / Chaikuad, A. / Dixon-Clarke, S.E. / Bullock, A.N. / Kopanchuk, S. / Ivan, T. / Ekambaram, R. / Viht, K. / Knapp, S. / Uri, A. |
External links | Molecules / PubMed:34299628 |
Methods | X-ray diffraction |
Resolution | 1.95 - 1.97 Å |
Structure data | PDB-7oov: PDB-7oow: PDB-7oox: |
Chemicals | ChemComp-SO4: ChemComp-EDO: ChemComp-HOH: ChemComp-MG: ChemComp-PO4: |
Source |
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Keywords | TRANSFERASE / PIM1 / inhibitor / kinase / kinase substrate / Structural Genomics / Structural Genomics Consortium / SGC |