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-Structure paper
Title | Small-molecule inhibition of METTL3 as a strategy against myeloid leukaemia. |
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Journal, issue, pages | Nature, Vol. 593, Page 597-601, Year 2021 |
Publish date | Mar 30, 2021 (structure data deposition date) |
Authors | Yankova, E. / Blackaby, W. / Albertella, M. / Rak, J. / De Braekeleer, E. / Tsagkogeorga, G. / Pilka, E.S. / Aspris, D. / Leggate, D. / Hendrick, A.G. ...Yankova, E. / Blackaby, W. / Albertella, M. / Rak, J. / De Braekeleer, E. / Tsagkogeorga, G. / Pilka, E.S. / Aspris, D. / Leggate, D. / Hendrick, A.G. / Webster, N.A. / Andrews, B. / Fosbeary, R. / Guest, P. / Irigoyen, N. / Eleftheriou, M. / Gozdecka, M. / Dias, J.M.L. / Bannister, A.J. / Vick, B. / Jeremias, I. / Vassiliou, G.S. / Rausch, O. / Tzelepis, K. / Kouzarides, T. |
External links | Nature / PubMed:33902106 |
Methods | X-ray diffraction |
Resolution | 3 Å |
Structure data | PDB-7o2i: |
Chemicals | ChemComp-V22: ChemComp-DMS: ChemComp-HOH: |
Source |
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Keywords | RNA BINDING PROTEIN / methyltransferase / SAM / inhibitor / m6A |