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-Structure paper
Title | A Conformation Selective Mode of Inhibiting SRC Improves Drug Efficacy and Tolerability. |
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Journal, issue, pages | Cancer Res., Vol. 81, Page 5438-5450, Year 2021 |
Publish date | Feb 8, 2021 (structure data deposition date) |
![]() | Temps, C. / Lietha, D. / Webb, E.R. / Li, X.F. / Dawson, J.C. / Muir, M. / Macleod, K.G. / Valero, T. / Munro, A.F. / Contreras-Montoya, R. ...Temps, C. / Lietha, D. / Webb, E.R. / Li, X.F. / Dawson, J.C. / Muir, M. / Macleod, K.G. / Valero, T. / Munro, A.F. / Contreras-Montoya, R. / Luque-Ortega, J.R. / Fraser, C. / Beetham, H. / Schoenherr, C. / Lopalco, M. / Arends, M.J. / Frame, M.C. / Qian, B.Z. / Brunton, V.G. / Carragher, N.O. / Unciti-Broceta, A. |
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Methods | X-ray diffraction |
Resolution | 1.5 Å |
Structure data | ![]() PDB-7ng7: |
Chemicals | ![]() ChemComp-EDO: ![]() ChemComp-UCW: ![]() ChemComp-HOH: |
Source |
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![]() | SIGNALING PROTEIN / Src kinase / inhibitor complex / inactive kinase |