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-Structure paper
Title | Antipsychotic phenothiazine drugs bind to KRAS in vitro. |
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Journal, issue, pages | J. Biomol. Nmr, Vol. 75, Page 233-244, Year 2021 |
Publish date | Jan 20, 2021 (structure data deposition date) |
![]() | Wang, X. / Gorfe, A.A. / Putkey, J.A. |
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Methods | NMR (solution) |
Structure data | ![]() PDB-7lgi: ![]() PDB-7mqu: |
Chemicals | ![]() ChemComp-GDP: ![]() ChemComp-MG: ![]() ChemComp-P2Z: ![]() ChemComp-ZM7: |
Source |
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![]() | HYDROLASE / GDP KRAS / SMALL MOLECULE LIGAND / HADDOCK STRUCTURE MODEL / CHEMICAL SHIFT CHANGES / INTERMOLECULAR NOE / HYDROLASE/HYDROLASE inhibitor / KRas / allosteric inhibitor / drug discovery / HADDOCK / HYDROLASE-HYDROLASE inhibitor complex |