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-Structure paper
Title | Synthesis and structural characterization of a monocarboxylic inhibitor for GRB2 SH2 domain. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 51, Page 128354-128354, Year 2021 |
Publish date | May 4, 2021 (structure data deposition date) |
Authors | Xiao, T. / Sun, L. / Zhang, M. / Li, Z. / Haura, E.B. / Schonbrunn, E. / Ji, H. |
External links | Bioorg. Med. Chem. Lett. / PubMed:34506932 |
Methods | X-ray diffraction |
Resolution | 2 Å |
Structure data | PDB-7mph: |
Chemicals | ChemComp-ZLY: ChemComp-EDO: ChemComp-SO4: ChemComp-HOH: |
Source |
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Keywords | PROTEIN BINDING / Inhibitor / Complex / growth factor receptor / Ras-MAPK signaling cascade |