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-Structure paper
Title | A kinase-cGAS cascade to synthesize a therapeutic STING activator. |
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Journal, issue, pages | Nature, Vol. 603, Page 439-444, Year 2022 |
Publish date | Apr 15, 2021 (structure data deposition date) |
![]() | McIntosh, J.A. / Liu, Z. / Andresen, B.M. / Marzijarani, N.S. / Moore, J.C. / Marshall, N.M. / Borra-Garske, M. / Obligacion, J.V. / Fier, P.S. / Peng, F. ...McIntosh, J.A. / Liu, Z. / Andresen, B.M. / Marzijarani, N.S. / Moore, J.C. / Marshall, N.M. / Borra-Garske, M. / Obligacion, J.V. / Fier, P.S. / Peng, F. / Forstater, J.H. / Winston, M.S. / An, C. / Chang, W. / Lim, J. / Huffman, M.A. / Miller, S.P. / Tsay, F.R. / Altman, M.D. / Lesburg, C.A. / Steinhuebel, D. / Trotter, B.W. / Cumming, J.N. / Northrup, A. / Bu, X. / Mann, B.F. / Biba, M. / Hiraga, K. / Murphy, G.S. / Kolev, J.N. / Makarewicz, A. / Pan, W. / Farasat, I. / Bade, R.S. / Stone, K. / Duan, D. / Alvizo, O. / Adpressa, D. / Guetschow, E. / Hoyt, E. / Regalado, E.L. / Castro, S. / Rivera, N. / Smith, J.P. / Wang, F. / Crespo, A. / Verma, D. / Axnanda, S. / Dance, Z.E.X. / Devine, P.N. / Tschaen, D. / Canada, K.A. / Bulger, P.G. / Sherry, B.D. / Truppo, M.D. / Ruck, R.T. / Campeau, L.C. / Bennett, D.J. / Humphrey, G.R. / Campos, K.R. / Maddess, M.L. |
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Methods | X-ray diffraction |
Resolution | 2.32 Å |
Structure data | ![]() PDB-7mhc: |
Chemicals | ![]() ChemComp-ZEV: ![]() ChemComp-HOH: |
Source |
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![]() | IMMUNE SYSTEM / STING / RECEPTOR / LIGAND COMPLEX / AGONIST / CLOSED CONFORMATION |