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| Title | Vimseltinib: A Precision CSF1R Therapy for Tenosynovial Giant Cell Tumors and Diseases Promoted by Macrophages. |
|---|---|
| Journal, issue, pages | Mol. Cancer Ther., Vol. 20, Page 2098-2109, Year 2021 |
| Publish date | Apr 8, 2021 (structure data deposition date) |
Authors | Smith, B.D. / Kaufman, M.D. / Wise, S.C. / Ahn, Y.M. / Caldwell, T.M. / Leary, C.B. / Lu, W.P. / Tan, G. / Vogeti, L. / Vogeti, S. ...Smith, B.D. / Kaufman, M.D. / Wise, S.C. / Ahn, Y.M. / Caldwell, T.M. / Leary, C.B. / Lu, W.P. / Tan, G. / Vogeti, L. / Vogeti, S. / Wilky, B.A. / Davis, L.E. / Sharma, M. / Ruiz-Soto, R. / Flynn, D.L. |
External links | Mol. Cancer Ther. / PubMed:34433663 |
| Methods | X-ray diffraction |
| Resolution | 2.8 Å |
| Structure data | ![]() PDB-7mfc: |
| Chemicals | ![]() ChemComp-Z6V: ![]() ChemComp-HOH: |
| Source |
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Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / cancer / TRANSFERASE-TRANSFERASE INHIBITOR complex |
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homo sapiens (human)
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