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-Structure paper
Title | Discovery of Soticlestat, a Potent and Selective Inhibitor for Cholesterol 24-Hydroxylase (CH24H). |
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Journal, issue, pages | J. Med. Chem., Vol. 64, Page 12228-12244, Year 2021 |
Publish date | Feb 16, 2021 (structure data deposition date) |
![]() | Koike, T. / Yoshikawa, M. / Ando, H.K. / Farnaby, W. / Nishi, T. / Watanabe, E. / Yano, J. / Miyamoto, M. / Kondo, S. / Ishii, T. / Kuroita, T. |
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Methods | X-ray diffraction |
Resolution | 1.995 - 2.15 Å |
Structure data | ![]() PDB-7lrl: ![]() PDB-7ls3: ![]() PDB-7ls4: |
Chemicals | ![]() ChemComp-HEM: ![]() ChemComp-YBS: ![]() ChemComp-HOH: ![]() ChemComp-YCJ: ![]() ChemComp-YCG: |
Source |
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![]() | HYDROLASE / cyp46a1 / ch24h / sbdd / drug discovery |