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-Structure paper
Title | Structure-Based Design of A-1293102, a Potent and Selective BCL-XL Inhibitor |
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Journal, issue, pages | ACS Medicinal Chemistry Letters, Vol. 12, Page 1011-1016, Year 2021 |
Publish date | Jan 21, 2021 (structure data deposition date) |
![]() | Tao, Z.F. / Wang, X. / Chen, J. / Ingram, J.P. / Jin, S. / Judge, R.A. / Kovar, P.J. / Park, C. / Sun, C. / Wakefield, B.D. ...Tao, Z.F. / Wang, X. / Chen, J. / Ingram, J.P. / Jin, S. / Judge, R.A. / Kovar, P.J. / Park, C. / Sun, C. / Wakefield, B.D. / Zhou, L. / Zhang, H. / Elmore, S.W. / Phillips, D.C. / Judd, A.S. / Leverson, J.D. / Souers, A.J. |
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Methods | X-ray diffraction |
Resolution | 1.409 Å |
Structure data | ![]() PDB-7lh7: |
Chemicals | ![]() ChemComp-XZM: ![]() ChemComp-HOH: |
Source |
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![]() | APOPTOSIS / Bcl-xL / structure-based drug design |