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-Structure paper
Title | Mobocertinib (TAK-788): A Targeted Inhibitor of EGFR Exon 20 Insertion Mutants in Non-Small Cell Lung Cancer. |
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Journal, issue, pages | Cancer Discov, Vol. 11, Page 1672-1687, Year 2021 |
Publish date | Jan 21, 2021 (structure data deposition date) |
![]() | Gonzalvez, F. / Vincent, S. / Baker, T.E. / Gould, A.E. / Li, S. / Wardwell, S.D. / Nadworny, S. / Ning, Y. / Zhang, S. / Huang, W.S. ...Gonzalvez, F. / Vincent, S. / Baker, T.E. / Gould, A.E. / Li, S. / Wardwell, S.D. / Nadworny, S. / Ning, Y. / Zhang, S. / Huang, W.S. / Hu, Y. / Li, F. / Greenfield, M.T. / Zech, S.G. / Das, B. / Narasimhan, N.I. / Clackson, T. / Dalgarno, D. / Shakespeare, W.C. / Fitzgerald, M. / Chouitar, J. / Griffin, R.J. / Liu, S. / Wong, K.K. / Zhu, X. / Rivera, V.M. |
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Methods | X-ray diffraction |
Resolution | 3.1 Å |
Structure data | ![]() PDB-7lgs: |
Chemicals | ![]() ChemComp-Q6K: ![]() ChemComp-EDO: ![]() ChemComp-CIT: ![]() ChemComp-HOH: |
Source |
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![]() | HYDROLASE/HYDROLASE inhibitor / Kinase / inhibitor / covalent / HYDROLASE / HYDROLASE-HYDROLASE inhibitor complex |