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-Structure paper
Title | Discovery of Selective Pituitary Adenylate Cyclase 1 Receptor (PAC1R) Antagonist Peptides Potent in a Maxadilan/PACAP38-Induced Increase in Blood Flow Pharmacodynamic Model. |
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Journal, issue, pages | J. Med. Chem., Vol. 64, Page 3427-3438, Year 2021 |
Publish date | Aug 10, 2020 (structure data deposition date) |
![]() | Hu, E. / Hong, F.T. / Aral, J. / Long, J. / Piper, D.E. / Poppe, L. / Andrews, K.L. / Hager, T. / Davis, C. / Li, H. ...Hu, E. / Hong, F.T. / Aral, J. / Long, J. / Piper, D.E. / Poppe, L. / Andrews, K.L. / Hager, T. / Davis, C. / Li, H. / Wong, P. / Gavva, N. / Shi, L. / Zhu, D.X.D. / Lehto, S.G. / Xu, C. / Miranda, L.P. |
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Methods | X-ray diffraction |
Resolution | 2.7 Å |
Structure data | ![]() PDB-7jqd: |
Chemicals | ![]() ChemComp-HOH: |
Source |
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![]() | SIGNALING PROTEIN/ANTAGONIST / ECD / Complex / Antagonist / GPCR / SIGNALING PROTEIN-ANTAGONIST complex |