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-Structure paper
Title | Discovery of a Series of Indane-Containing NBTIs with Activity against Multidrug-Resistant Gram-Negative Pathogens. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 14, Page 993-998, Year 2023 |
Publish date | Apr 18, 2023 (structure data deposition date) |
Authors | Cumming, J.G. / Kreis, L. / Kuhne, H. / Wermuth, R. / Vercruysse, M. / Kramer, C. / Rudolph, M.G. / Xu, Z. |
External links | Acs Med. Chem. Lett. / PubMed:37465290 |
Methods | X-ray diffraction |
Resolution | 2.081 - 2.16 Å |
Structure data | PDB-7fvs: PDB-7fvt: |
Chemicals | ChemComp-MN: ChemComp-CL: ChemComp-ACT: ChemComp-61I: ChemComp-HOH: ChemComp-6I0: |
Source |
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Keywords | ISOMERASE / DNA GYRASE / TOPOISOMERASE; |