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-Structure paper
Title | The X-ray structure of tubulysin analogue TGL in complex with tubulin and three possible routes for the development of next-generation tubulysin analogues. |
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Journal, issue, pages | Biochem. Biophys. Res. Commun., Vol. 565, Page 29-35, Year 2021 |
Publish date | Apr 15, 2021 (structure data deposition date) |
Authors | Li, W. / Tan, L. / Zhang, Z. / Xia, Q. / Lei, D. / Li, Y. / Zhang, T. / Zeng, S. / Sima, X. / Wang, Y. |
External links | Biochem. Biophys. Res. Commun. / PubMed:34090207 |
Methods | X-ray diffraction |
Resolution | 2.643 Å |
Structure data | PDB-7en3: |
Chemicals | ChemComp-GTP: ChemComp-MG: ChemComp-CA: ChemComp-GDP: ChemComp-MES: ChemComp-J6R: ChemComp-ACP: ChemComp-HOH: |
Source |
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Keywords | STRUCTURAL PROTEIN/INHIBITOR / microtubule assembly inhibitors / STRUCTURAL PROTEIN-INHIBITOR complex |