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-Structure paper
Title | Development of potent and selective inhibitors targeting the papain-like protease of SARS-CoV-2. |
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Journal, issue, pages | Cell Chem Biol, Vol. 28, Page 855-865.e9, Year 2021 |
Publish date | Sep 30, 2020 (structure data deposition date) |
Authors | Shan, H. / Liu, J. / Shen, J. / Dai, J. / Xu, G. / Lu, K. / Han, C. / Wang, Y. / Xu, X. / Tong, Y. ...Shan, H. / Liu, J. / Shen, J. / Dai, J. / Xu, G. / Lu, K. / Han, C. / Wang, Y. / Xu, X. / Tong, Y. / Xiang, H. / Ai, Z. / Zhuang, G. / Hu, J. / Zhang, Z. / Li, Y. / Pan, L. / Tan, L. |
External links | Cell Chem Biol / PubMed:33979649 |
Methods | X-ray diffraction |
Resolution | 1.6 - 2.4 Å |
Structure data | PDB-7d6h: PDB-7e35: |
Chemicals | ChemComp-ZN: ChemComp-PO4: ChemComp-HOH: ChemComp-GYX: |
Source |
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Keywords | HYDROLASE / Protease / Deubiquitinase / VIRAL PROTEIN / HYDROLASE/HYDROLASE INHIBITOR / HYDROLASE-HYDROLASE INHIBITOR complex |