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-Structure paper
Title | Identification of pyrogallol as a warhead in design of covalent inhibitors for the SARS-CoV-2 3CL protease. |
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Journal, issue, pages | Nat Commun, Vol. 12, Page 3623-3623, Year 2021 |
Publish date | Dec 21, 2020 (structure data deposition date) |
![]() | Su, H. / Yao, S. / Zhao, W. / Zhang, Y. / Liu, J. / Shao, Q. / Wang, Q. / Li, M. / Xie, H. / Shang, W. ...Su, H. / Yao, S. / Zhao, W. / Zhang, Y. / Liu, J. / Shao, Q. / Wang, Q. / Li, M. / Xie, H. / Shang, W. / Ke, C. / Feng, L. / Jiang, X. / Shen, J. / Xiao, G. / Jiang, H. / Zhang, L. / Ye, Y. / Xu, Y. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.75 - 2.35 Å |
Structure data | ![]() PDB-7dpp: ![]() PDB-7dpu: ![]() PDB-7dpv: |
Chemicals | ![]() ChemComp-MYC: ![]() ChemComp-HOH: ![]() ChemComp-HER: ![]() ChemComp-GOL: ![]() ChemComp-HF0: |
Source |
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![]() | VIRAL PROTEIN / SARS-CoV-2 / 3CLpro / inhibitor / complex / myricetin |