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Title | Design, Synthesis, and Biological Evaluation of Peptidomimetic Aldehydes as Broad-Spectrum Inhibitors against Enterovirus and SARS-CoV-2. |
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Journal, issue, pages | J. Med. Chem., Vol. 65, Page 2794-2808, Year 2022 |
Publish date | Dec 9, 2020 (structure data deposition date) |
Authors | Dai, W. / Jochmans, D. / Xie, H. / Yang, H. / Li, J. / Su, H. / Chang, D. / Wang, J. / Peng, J. / Zhu, L. ...Dai, W. / Jochmans, D. / Xie, H. / Yang, H. / Li, J. / Su, H. / Chang, D. / Wang, J. / Peng, J. / Zhu, L. / Nian, Y. / Hilgenfeld, R. / Jiang, H. / Chen, K. / Zhang, L. / Xu, Y. / Neyts, J. / Liu, H. |
External links | J. Med. Chem. / PubMed:33872498 |
Methods | X-ray diffraction |
Resolution | 1.17 Å |
Structure data | PDB-7dnc: |
Chemicals | ChemComp-FHR: ChemComp-HOH: |
Source |
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Keywords | HYDROLASE / 3Cpro / inhibitor / complex |