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-Structure paper
Title | Discovery of selective BPTF bromodomain inhibitors by screening and structure-based optimization. |
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Journal, issue, pages | Biochem. Biophys. Res. Commun., Vol. 545, Page 125-131, Year 2021 |
Publish date | Dec 8, 2020 (structure data deposition date) |
![]() | Xiong, L. / Mao, X. / Guo, Y. / Zhou, Y. / Chen, M. / Chen, P. / Yang, S. / Li, L. |
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Methods | X-ray diffraction |
Resolution | 2 - 2.841 Å |
Structure data | ![]() PDB-7dmy: ![]() PDB-7dn4: |
Chemicals | ![]() ChemComp-HAF: ![]() ChemComp-HOH: ![]() ChemComp-JC3: |
Source |
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![]() | PROTEIN BINDING / inhibitor;BPTF;Bromodomain / inhibitor / BPTF / bromodomain / reader |