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-Structure paper
Title | Structure-Based Identification of Potent Lysine-Specific Demethylase 1 Inhibitor Peptides and Temporary Cyclization to Enhance Proteolytic Stability and Cell Growth-Inhibitory Activity. |
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Journal, issue, pages | J. Med. Chem., Vol. 64, Page 3707-3719, Year 2021 |
Publish date | Jun 19, 2020 (structure data deposition date) |
![]() | Kitagawa, H. / Kikuchi, M. / Sato, S. / Watanabe, H. / Umezawa, N. / Kato, M. / Hisamatsu, Y. / Umehara, T. / Higuchi, T. |
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Methods | X-ray diffraction |
Resolution | 2.64 - 2.8 Å |
Structure data | ![]() PDB-7cdc: ![]() PDB-7cdd: ![]() PDB-7cde: ![]() PDB-7cdf: ![]() PDB-7cdg: |
Chemicals | ![]() ChemComp-FAD: ![]() ChemComp-GOL: ![]() ChemComp-HOH: |
Source |
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![]() | OXIDOREDUCTASE/TRANSCRIPTION / DEMETHYLASE / AMINE OXIDASE / CHROMATIN / HISTONE / FAD / COREPRESSOR / OXIDOREDUCTASE-TRANSCRIPTION-INHIBITOR complex / OXIDOREDUCTASE / OXIDOREDUCTASE-TRANSCRIPTION complex |